产品名 | |||
Pimasertib (AS-703026) | MEK | 卵巢癌,黑色素瘤 | Phase 2 |
MLN2480 | Raf | 黑色素瘤 | Phase 1 |
RG7304 | MEK | 实体瘤,骨髓瘤 | Phase 1 |
GDC-0994 | ERK | 实体瘤 | Phase 1 |
Peficitinib (ASP015K, JNJ-54781532) | JAK | 类风湿性关节炎 | Phase 3 |
LY2784544 | JAK | 骨髓增生性疾病 | Phase 2 |
Filgotinib (GLPG0634) | JAK | 类风湿性关节炎,克罗恩病 | Phase 2 |
Losmapimod (GW856553X) | p38 MAPK | 急性冠脉综合征 | Phase 3 |
SB-681323 | p38 MAPK | 类风湿性关节炎,神经性疼痛,冠状动脉疾病,阻塞性肺疾病 | Phase 2 |
PH-797804 | p38 MAPK | 阻塞性肺疾病,带状疱疹后神经痛,类风湿性关节炎 | Phase 2 |
Tak-715 | p38 MAPK | 类风湿性关节炎 | Phase 2 |
BMS-582949 | p38 MAPK | 类风湿性关节炎 | Phase 2 |
Fostamatinib (R788) | Syk | 血小板减少性紫癜 | Phase 3 |
Entospletinib (GS-9973) | Syk | 淋巴瘤,白血病 | Phase 2 |
PRT062607 (P505-15, BIIB057) HCl | Syk | 类风湿关节炎,狼疮 | Phase 2 |
Trelagliptin (SYR-472) | DPP-4 | 糖尿病 | Phase 3 |
Omarigliptin (MK-3102) | DPP-4 | 糖尿病 | Phase 3 |
Asunaprevir (BMS-650032) | HCV Protease | HCV感染 | Phase 3 |
Faldaprevir (BI 201335) | HCV Protease | HCV感染 | Phase 3 |
Vaniprevir (MK-7009) | HCV Protease | HCV感染 | Phase 3 |
Danoprevir (ITMN-191) | HCV Protease | HCV感染 | Phase 2 |
GS-9451 | HCV Protease | HCV感染 | Phase 2 |
GS-9669 | HCV Protease | HCV感染 | Phase 2 |