| 产品名 | |||
| Carfilzomib (PR-171) | Proteasome | 骨髓瘤 | 2012/7/20 |
| Ivacaftor (VX-770) | CFTR | 囊性纤维化 | 2012/1/31 |
| Vismodegib (GDC-0449) | Hedgehog/Smoothened | 基底细胞癌 | 2012/1/30 |
| Axitinib | VEGFR | 肾细胞癌 | 2012/1/27 |
| Ruxolitinib (INCB018424) | JAK | 骨髓纤维化 | 2011/11/16 |
| Crizotinib (PF-02341066) | c-Met | 肺癌 | 2011/8/26 |
| Vemurafenib (PLX4032, RG7204) | Raf | 黑色素瘤 | 2011/8/17 |
| Docetaxel | Microtubule Associated | 乳腺癌,肺癌,胃癌,头颈癌,前列腺癌 | 2011/5/3 |
| Abiraterone Acetate | P450 (e.g. CYP17) | 前列腺癌 | 2011/4/28 |
| Vandetanib (ZD6474) | VEGFR | 甲状腺癌 | 2011/4/6 |
| Roflumilast | PDE | 哮喘,肺病 | 2011/2/28 |
| Topotecan HCl | Topoisomerase | 肺癌,卵巢癌,子宫颈癌 | 2011/2/25 |
| Gemcitabine HCl | DNA/RNA Synthesis | 淋巴瘤,肺癌,尿道上皮癌,乳腺癌,卵巢癌,胆管癌,胰腺癌 | 2011/1/25 |
| Fingolimod (FTY720) HCl | S1P Receptor | 多发性硬化 | 2010/9/21 |
| Romidepsin (FK228, Depsipeptide) | HDAC | 淋巴瘤 | 2009/11/5 |
| Everolimus (RAD001) | mTOR | 肾细胞癌,乳腺癌,胰腺癌,结节性硬化症综合征 | 2009/4/30 |
| Bicalutamide | Androgen Receptor | 前列腺癌 | 2008/12/19 |
| Plerixafor 8HCl (AMD3100 8HCl) | CXCR | 淋巴瘤,骨髓瘤 | 2008/12/15 |
| Nilotinib (AMN-107) | Bcr-Abl | 白血病 | 2007/10/29 |
| Raltegravir (MK-0518) | Integrase | 艾滋病毒感染 | 2007/10/12 |
| Maraviroc | CCR | 艾滋病毒感染 | 2007/8/6 |
| Rapamycin (Sirolimus) | mTOR | 淋巴瘤 | 2007/5/30 |
| Temsirolimus (CCI-779, NSC 683864) | mTOR | 肾细胞癌,淋巴瘤 | 2007/5/30 |
